SCHEMBL27488641

SCHEMBL27488641

O=COCCc1ccsc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.48
HPGD P15428 2/20 0.43
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MEN1 O00255 1/20 0.34
KDM4A O75164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5535967 0.89 TAAR1 (0.46) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL5541802 0.87 TAAR1 (0.44) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL5541464 0.86 TAAR1 (0.43) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL5544151 0.86 TAAR1 (0.43) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL7686942 0.81 TAAR1 (0.48) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL5541959 0.80
SCHEMBL29009267 0.79 TAAR1 (0.47) TAAR1HPGDDRD2DRD3SLC1A3
Hydrochloric Acid SCHEMBL28198042 0.78 SLC1A3 (0.46) TAAR1HPGDDRD2DRD3SLC1A3
SCHEMBL25386744 0.74
SCHEMBL8256108 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109912621-A A kind of asymmetric naphthalene core small molecule receptor material and its preparation method and application 湖南科技大学 2019-06-21 CN claimed
CN-109776567-A A kind of hexa-atomic bridged ring pyrene core small molecule receptor material and its preparation method and application 湖南科技大学 2019-05-21 CN claimed
CN-109776568-A Axisymmetric hexa-atomic bridged ring naphthalene core small molecule receptor material of one kind and its preparation method and application 湖南科技大学 2019-05-21 CN claimed
CN-104703992-B Process for preparing thienopyrimidine derivatives 武田药品工业株式会社 2019-03-05 CN claimed
CN-109053766-A The preparation method of Thienopyrimidine derivative 武田药品工业株式会社 2018-12-21 CN claimed
CN-106366095-A Polycyclic-based field effect transistor material and preparation method and application thereof 苏州大学 2017-02-01 CN claimed
CN-102924429-B 1,2-naphthaquinone derivatives and preparation method thereof UNIV XINXIANG MEDICAL 2013-12-11 CN claimed
CN-103242290-A Preparation method of 6-tert-butyl-4,5,6,7-tetrahydrobenzothiophene-2-amine KEJIE BIO SUZHOU PHARMACEUTICAL CO LTD 2013-08-14 CN claimed
CN-102924429-A 1,2-naphthaquinone derivatives and preparation method thereof UNIV XINXIANG MEDICAL 2013-02-13 CN claimed
CN-101857588-A 4-aromatic aminoquinazoline derivative and purpose thereof UNIV SOUTHEAST 2010-10-13 CN claimed
CN-110475776-A For preventing and treating the tricyclic carboxylic acid amides of arthropod BAYER CROPSCIENCE AG 2019-11-19 CN disclosed
CN-110115365-A The adjusting that actinism receptor and relative ligand are carried out 西诺米克斯公司 2019-08-13 CN disclosed
CN-109970760-A ACC inhibitor and its purposes 吉利德阿波罗公司 2019-07-05 CN disclosed
CN-109912621-A A kind of asymmetric naphthalene core small molecule receptor material and its preparation method and application 湖南科技大学 2019-06-21 CN disclosed
CN-106905346-B ACC inhibitor and its purposes 吉利德阿波罗公司 2019-05-28 CN disclosed
CN-1522258-A Novel 4-amino-5, 6-substituted thieno [2, 3-D ] pyrimidine compounds 2004-08-18 CN disclosed
CN-1489458-A Inflammatory cytokine production dissociation inhibitor ��ʽ����ҽҩ��������о��� 2004-04-14 CN disclosed
CN-1422265-A Process for producing benzo-fused heterocycle MERCK PATENT GMBH (DE) 2003-06-04 CN disclosed
CN-1335777-A Preventives or remedies for myocarditis, dilated cardiomyopathy and cardiac insufficiency containing NF-K B inhibitors as the active ingredient SUNTORY LTD (JP) 2002-02-13 CN disclosed
CN-1228701-A Heterocyclic compounds with thrombolytic activity and their use for treating thrombosis DUPIN JEAN PIERRE (FR) 1999-09-15 CN disclosed