SCHEMBL27497487

SCHEMBL27497487

Cc1nc(C(=O)OC(C)(C)C)c(C)c(N)c1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
ALDH1A1 P00352 5/20 0.33
HPGD P15428 2/20 0.33
CYP1A2 P05177 1/20 0.32
LMNA P02545 1/20 0.31
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31
DHFR P00374 1/20 0.31
KDM4E B2RXH2 2/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27497162 0.86 GRM6 (0.35) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL27961512 0.72 CYP2C9 (0.40) GRM6CYP2C9CYP2C19NPSR1CNR1
Methane SCHEMBL27512739 0.72 GRM6 (0.36) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL19625997 0.71 NPSR1 (0.52) NPSR1ALDH1A1HPGDKDM4EGAA
SCHEMBL6977590 0.69 CFTR (0.36) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL7385332 0.69 CFTR (0.36) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL3963821 0.69 MEN1 (0.39) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL6985283 0.69 ALDH1A1 (0.53) GRM6ALDH1A1HPGDCYP1A2LMNA
SCHEMBL14634345 0.68 GRM5 (0.47) GRM6CYP2C9CYP2C19NPSR1CNR1
SCHEMBL5556257 0.67 GRM6 (0.40) GRM6CYP2C9CYP2C19NPSR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1222909-A Pyrazinone thrombin inhibitors MERCK & CO INC (US) 1999-07-14 CN disclosed