SCHEMBL27503243

SCHEMBL27503243

Cn1cccc(-c2ccc(C[C@H](N)C(=O)O)cc2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.54
ITGA4 P13612 3/20 0.54
ITGB7 P26010 2/20 0.54
SLC7A5 Q01650 3/20 0.50
PTGS1 P23219 2/20 0.50
ALPI P09923 1/20 0.50
PKM P14618 1/20 0.50
XIAP P98170 1/20 0.50
TYR P14679 5/20 0.45
GRB2 P62993 1/20 0.45
TPH1 P17752 6/20 0.43
PTPN1 P18031 1/20 0.42
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
EGFR P00533 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27503244 1.00 ITGB1 (0.54) ITGB1ITGA4ITGB7SLC7A5PTGS1
SCHEMBL6236132 0.86 ITGA4 (0.51) ITGB1ITGA4ITGB7PTGS2
SCHEMBL27522587 0.86 ITGA4 (0.51) ITGB1ITGA4ITGB7PTGS2
Hydrochloric Acid SCHEMBL27489194 0.85 ITGA4 (0.50) ITGB1ITGA4ITGB7TPH1PTGS2
Hydrochloric Acid SCHEMBL6236128 0.85 ITGA4 (0.50) ITGB1ITGA4ITGB7TPH1PTGS2
SCHEMBL25146739 0.80 ITGB1 (0.49) ITGB1ITGA4ITGB7PTGS1KDM4E
SCHEMBL27488546 0.79 ITGB1 (0.59) ITGB1ITGA4ITGB7SLC7A5PTGS1
SCHEMBL27488545 0.79 ITGB1 (0.59) ITGB1ITGA4ITGB7SLC7A5PTGS1
SCHEMBL180446 0.78 SLC7A5 (0.70) SLC7A5PTGS1ALPIPKMXIAP
SCHEMBL27494301 0.78 SLC7A5 (0.50) ITGB1ITGA4ITGB7SLC7A5PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1196682-C 4-pyridyl-N-acyl-L-phenylalanine HOFFMANN LA ROCHE (CH) 2005-04-13 CN disclosed
CN-1402709-A 4-pyridinyl-N-acyl-L-phenylalanines HOFFMANN LA ROCHE (CH) 2003-03-12 CN disclosed