SCHEMBL27510491

SCHEMBL27510491

CN1c2ccc(Br)cc2C(c2ccccc2F)=NC(C(=O)OCc2ccccc2)C1N

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 8/20 0.42
CCKAR P32238 4/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27533179 0.82 CCKBR (0.40) CCKBRCCKARCYP2C9CYP2C19
SCHEMBL27528202 0.79 CCKBR (0.42) CCKBRCCKARCYP2C9CYP2C19GABRA1
SCHEMBL4424638 0.79 CCKBR (0.44) CCKBRCCKARCYP2C9CYP2C19
SCHEMBL27510203 0.77 CCKBR (0.47) CCKBRCCKAR
SCHEMBL4413353 0.76 CCKBR (0.60) CCKBRCCKAR
SCHEMBL27510490 0.76 CCKBR (0.49) CCKBRCCKAR
SCHEMBL4413355 0.73 CYP2C9 (0.39) CCKBRCCKARCYP2C9CYP2C19GABRA1
SCHEMBL11961451 0.71 BRD4 (0.68) CCKBR
SCHEMBL27528231 0.71 CCKBR (0.42) CCKBRCCKARCYP2C9CYP2C19GABRA1
SCHEMBL27587107 0.70 CYP3A4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1242007-A Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising such compounds, and methods of inhibiting beta amyloid peptide release and/or its synthesis using such compounds ELAND PHARMACEUTICAL CORP (US) 2000-01-19 CN disclosed