SCHEMBL27528331

SCHEMBL27528331

NCc1ccc(CN2CCN(c3ccc4ccccc4n3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.62
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 4/20 0.55
HTR3A P46098 3/20 0.55
HTR3E A5X5Y0 2/20 0.55
HTR3B O95264 2/20 0.55
CYP1A2 P05177 2/20 0.55
HTR3D Q70Z44 2/20 0.55
HTR3C Q8WXA8 2/20 0.55
THPO P40225 1/20 0.55
HRH4 Q9H3N8 1/20 0.55
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
HTR1A P08908 4/20 0.51
TDP1 Q9NUW8 2/20 0.51
USP2 O75604 1/20 0.51
ADRB1 P08588 1/20 0.51
CYP3A4 P08684 1/20 0.51
HTR2C P28335 1/20 0.51
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27494769 0.99 HRH3 (0.60) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6231596 0.89 HRH3 (0.68) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6229963 0.88 HRH3 (0.63) HRH3KDM4EALDH1A1HTR3AHTR3E
Bromide SCHEMBL6232431 0.86 HRH3 (0.62) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6232468 0.86 HRH3 (0.66) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6229177 0.86 HRH3 (0.62) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6228769 0.86 HRH3 (0.70) HRH3KDM4EALDH1A1HTR3AHTR3E
Hydrochloric Acid SCHEMBL6234227 0.85 HRH3 (0.64) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6229805 0.83 CASP1 (0.58) HRH3KDM4EALDH1A1HTR3AHTR3E
SCHEMBL6230285 0.83 HRH3 (0.61) HRH3KDM4EALDH1A1HTR3AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1283195-A 1-(2-naphthyl) and 1(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine D4 receptor subtype ligands NEUROGEN CORP (US) 2001-02-07 CN claimed