SCHEMBL27544429

SCHEMBL27544429

CC(=O)Oc1nc(-c2ccccc2)cnc1N

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 15/20 0.50
PRKDC P78527 6/20 0.50
ALOX5 P09917 1/20 0.47
NEK2 P51955 1/20 0.45
LDHA P00338 1/20 0.43
LDHB P07195 1/20 0.43
ATM Q13315 2/20 0.43
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27836947 0.87 ATR (0.54) ATR
SCHEMBL27912649 0.81 ATR (0.50) ATRAURKAAURKB
SCHEMBL27836793 0.80 ACVR1 (0.42) ATRPRKDC
SCHEMBL2581392 0.80 MAPT (0.51) ATRPRKDCATM
SCHEMBL3459860 0.79 ATR (0.46) ATRPRKDCNEK2ATM
SCHEMBL14525246 0.77 ATR (0.65) ATRPRKDCATM
SCHEMBL935340 0.75 AURKA (0.48) ATRPRKDCAURKAAURKB
SCHEMBL3462566 0.75 ATR (0.66) ATRPRKDCATM
SCHEMBL28944517 0.74 GRM5 (0.39) ALOX5
SCHEMBL27517890 0.74 ATR (0.39) ATRALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1280289-C Alkoxy carbonylamino heteroaryl carboxylic acid derivatives as IP antagonists HOFFMANN LA ROCHE (CH) 2006-10-18 CN disclosed
CN-1494544-A Alkoxy carbonylamino heteroaryl carboxylic acid derivatives as IP antagonists - 2004-05-05 CN disclosed