SCHEMBL27547005

SCHEMBL27547005

COc1c(F)c(Cl)c(F)c(C=O)c1F

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.33
ALDH1A1 P00352 1/20 0.31
ERN1 O75460 3/20 0.31
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27257037 0.84 IMPDH2 (0.30) IMPDH2ERN1
SCHEMBL28165391 0.81 ERN1 (0.33) ALDH1A1ERN1
SCHEMBL18241122 0.81 ERN1 (0.35) ALDH1A1ERN1AKR1B1
SCHEMBL6568843 0.79 HSD17B10 (0.32) ALDH1A1ERN1AKR1B1
SCHEMBL1810542 0.78 MEN1 (0.36) ALDH1A1
SCHEMBL6060779 0.78 MEN1 (0.36) ALDH1A1
SCHEMBL27893581 0.76 MEN1 (0.31) IMPDH2ALDH1A1ERN1
SCHEMBL11017584 0.73 HSD17B10 (0.33)
SCHEMBL31335743 0.73 ERN1 (0.43) ALDH1A1ERN1
SCHEMBL28056767 0.72 ERN1 (0.36) ALDH1A1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1939903-A Mandelic acid derivatives and their use as throbin inhibitors ASTRAZENECA AB (SE) 2007-04-04 CN disclosed
CN-1939902-A Mandelic acid derivatives and their use as throbin inhibitors ASTRAZENECA AB (SE) 2007-04-04 CN disclosed
CN-1291975-C Novel mandelic acid derivatives and their use as thrombin inhibitors ASTRAZENECA AB (SE) 2006-12-27 CN disclosed
CN-1656066-A combination drug ASTRAZENECA AB (SE) 2005-08-17 CN disclosed
CN-1487919-A Novel mandelic acid derivatives and their use as thrombin inhibitors 2004-04-07 CN disclosed