SCHEMBL27558441

SCHEMBL27558441

CC(NC(=O)c1ncc[nH]1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 1/20 0.50
KDM4C Q9H3R0 1/20 0.47
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
EGLN1 Q9GZT9 4/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CA2 P00918 2/20 0.39
CA1 P00915 2/20 0.39
AKR1B1 P15121 2/20 0.39
HDAC4 P56524 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
BBOX1 O75936 2/20 0.37
FTO Q9C0B1 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1509747 1.00 HSPA5 (0.50) HSPA5KDM4CNPC1RAB9AEGLN1
SCHEMBL12724861 0.84 HSPA5 (0.53) HSPA5NPC1RAB9AKMT2AALDH1A1
SCHEMBL1509778 0.79 MAPT (0.49) HSPA5KMT2AMEN1ALDH1A1
SCHEMBL27460343 0.79 HSPA5 (0.40) HSPA5KDM4CNPC1RAB9A
SCHEMBL8645316 0.79 HSPA5 (0.40) HSPA5KDM4CNPC1RAB9A
SCHEMBL8890777 0.79 HSPA5 (0.49) HSPA5NPC1RAB9AKMT2AMEN1
SCHEMBL8890772 0.79 HSPA5 (0.49) HSPA5NPC1RAB9AKMT2AMEN1
SCHEMBL11142669 0.78 HSPA5 (0.48) HSPA5NPC1RAB9AKMT2A
SCHEMBL12450657 0.77 HSPA5 (0.48) HSPA5NPC1RAB9A
SCHEMBL27460341 0.77 HSPA5 (0.41) HSPA5NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1980658-A Treatment of diseases using ICE inhibitors VERTEX PHARMA (US) 2007-06-13 CN disclosed
CN-1298707-C Imidazole and benzimidazole caspase inhibitors and uses thereof VERTEX PHARMA INC (US) 2007-02-07 CN disclosed
CN-1481367-A Imidazole and benzimiddzole caspase inhibitors and uses thereof ��̩��˹ҩ��ɷ����޹�˾ 2004-03-10 CN disclosed