SCHEMBL27563151

SCHEMBL27563151

COC(=O)C(F)c1c[nH]c2cnccc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 9/20 0.40
GSK3B P49841 5/20 0.40
NFATC1 O95644 5/20 0.40
CDK2 P24941 3/20 0.39
DYRK1B Q9Y463 3/20 0.39
PDPK1 O15530 1/20 0.39
TGFBR1 P36897 1/20 0.39
IKBKE Q14164 1/20 0.39
KDM5A P29375 2/20 0.38
KDM5B Q9UGL1 1/20 0.38
GPR84 Q9NQS5 2/20 0.37
IGF1R P08069 1/20 0.37
NR4A2 P43354 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
CPT1A P50416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27583278 0.89 NR4A2 (0.39) DYRK1AGSK3BDYRK1BNR4A2KDR
SCHEMBL27563134 0.77 MAP2K1 (0.56) DYRK1AGSK3BCDK2GPR84
SCHEMBL20904626 0.74 NR4A2 (0.40) DYRK1AGSK3BDYRK1BNR4A2KDR
SCHEMBL27583279 0.74 DYRK1A (0.35) DYRK1AKDM5ANR4A2
SCHEMBL12491378 0.73 DYRK1A (0.49) DYRK1AGSK3BNFATC1CDK2DYRK1B
SCHEMBL27583266 0.73 MAP2K1 (0.39) GSK3BNR4A2KDRFLT3
SCHEMBL6780792 0.73 TACR1 (0.47) DYRK1AGSK3BCDK2DYRK1BGPR84
SCHEMBL2611046 0.73 DYRK1A (0.51) DYRK1AGSK3BNFATC1CDK2DYRK1B
SCHEMBL1607800 0.73 NR4A2 (0.62) DYRK1AGSK3BNR4A2CPT1A
SCHEMBL31753965 0.73 NR4A2 (0.62) DYRK1AGSK3BNR4A2CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1404392-A Antiviral azaindole derivatives BRISTOL MYERS SQUIBB CO (US) 2003-03-19 CN disclosed