SCHEMBL27564366

SCHEMBL27564366

Cc1[nH]ccc1C1C(=O)Nc2ccc(S(=O)(=O)NCCO)cc21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
ALDH1A1 P00352 3/20 0.43
PKM P14618 3/20 0.43
GAA P10253 1/20 0.43
POLB P06746 3/20 0.43
ILK Q13418 1/20 0.40
NEK1 Q96PY6 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
THRB P10828 1/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP2C19 P33261 2/20 0.36
BRD4 O60885 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27582058 0.84 MAPT (0.41) MAPTALDH1A1PKMGAAPOLB
SCHEMBL28749800 0.84 MAPK1 (0.47) MAPTALDH1A1GAANEK1LMNA
SCHEMBL28747307 0.82 ALDH1A1 (0.54) ALDH1A1PKMPOLBILKNEK1
SCHEMBL27581877 0.81 CA1 (0.41) MAPTALDH1A1PKMMEN1KMT2A
SCHEMBL27564363 0.78 ALDH1A1 (0.37) MAPTALDH1A1PKMGAAPOLB
SCHEMBL13698175 0.78 ALDH1A1 (0.49) MAPTALDH1A1PKMGAAPOLB
SCHEMBL13698113 0.77 ALDH1A1 (0.48) MAPTALDH1A1PKMGAAPOLB
SCHEMBL27561520 0.74 PDPK1 (0.41) ALDH1A1IKBKBCHUKBRD4
SCHEMBL27582054 0.72 DDB1 (0.33) POLBTP53BRD4
SCHEMBL27561502 0.72 KDM4E (0.56) MAPTALDH1A1GAALMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1351498-A Pyrrolotriazines inhibitors of kinases BRISTOL MYERS SQUIBB CO (US) 2002-05-29 CN disclosed