SCHEMBL27600166

SCHEMBL27600166

CCn1c(=O)c2c(nc(Cl)n2CCc2ccccc2)n(CC)c1=O

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.66
SIRT1 Q96EB6 1/20 0.54
SIRT3 Q9NTG7 1/20 0.54
SIRT5 Q9NXA8 1/20 0.54
ADORA2A P29274 3/20 0.53
ADORA3 P0DMS8 1/20 0.53
PDE5A O76074 2/20 0.53
LMNA P02545 1/20 0.50
TSHR P16473 1/20 0.50
CNOT7 Q9UIV1 1/20 0.49
ADORA2B P29275 2/20 0.48
POLB P06746 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27600387 0.91 LMNA (0.58) ADORA1SIRT1SIRT3SIRT5LMNA
SCHEMBL555828 0.88 ADORA1 (0.63) ADORA1ADORA2AADORA3PDE5AADORA2B
SCHEMBL27600589 0.87 LMNA (0.62) LMNATSHRPOLBHIF1A
SCHEMBL1947774 0.86 MAPT (0.54) ADORA1ADORA2AADORA3PDE5ALMNA
SCHEMBL27582891 0.85 LMNA (0.57) ADORA2AADORA3LMNATSHRADORA2B
SCHEMBL28749929 0.85 HIF1A (0.62) ADORA3LMNATSHRADORA2BPOLB
SCHEMBL555395 0.82 HTT (0.60) LMNATSHRPOLBHIF1A
SCHEMBL27582885 0.82 LMNA (0.73) LMNATSHR
SCHEMBL27600370 0.82 LMNA (0.57) LMNATSHR
SCHEMBL27583016 0.82 CYP1A2 (0.58) LMNATSHRCNOT7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed