SCHEMBL2760025

SCHEMBL2760025

CCCCOC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCc1ccccc1)NC(C)=O)[C@@H](C)OC(=O)OCOP=O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CPA1 P15085 2/20 0.42
CPA2 P48052 2/20 0.42
CPA4 Q9UI42 2/20 0.42
PSMB5 P28074 2/20 0.41
MMP3 P08254 5/20 0.40
MMP9 P14780 1/20 0.40
CTSL P07711 3/20 0.39
MMP2 P08253 2/20 0.39
CTSK P43235 1/20 0.39
MMP1 P03956 1/20 0.39
MMP12 P39900 1/20 0.39
MMP13 P45452 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CTSB P07858 1/20 0.37
REN P00797 1/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14208821 0.90 CTSL (0.47) CPA1CPA2CPA4MMP3CTSL
SCHEMBL2760023 0.89 CPA1 (0.48) CPA1CPA2CPA4MMP3CTSL
SCHEMBL2632751 0.89 CPA1 (0.44) CPA1CPA2CPA4PSMB5MMP3
SCHEMBL8270598 0.89 CPA1 (0.47) CPA1CPA2CPA4PSMB5MMP3
SCHEMBL2632750 0.88 CPA1 (0.41) CPA1CPA2CPA4PSMB5MMP3
SCHEMBL2632715 0.85 CPA1 (0.49) CPA1CPA2CPA4PSMB5MMP3
SCHEMBL2735653 0.82 PSMB5 (0.52) PSMB5CTSB
SCHEMBL2632731 0.81 CPA1 (0.50) CPA1CPA2CPA4PSMB5MMP3
SCHEMBL14208668 0.79 CTSL (0.49) CPA1CPA2CPA4MMP3CTSL
SCHEMBL2632733 0.79 CPA1 (0.47) CPA1CPA2CPA4PSMB5MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088741-B2 Compounds for enzyme inhibition ONYX THERAPEUTICS, INC. (US) 2012-01-03 US disclosed