SCHEMBL27611541

SCHEMBL27611541

CC(=O)OCn1ncc2ccc(N)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
CSNK1A1 P48729 1/20 0.47
GSK3A P49840 1/20 0.47
LIMK1 P53667 1/20 0.47
IKBKE Q14164 1/20 0.47
MAPK14 Q16539 1/20 0.47
TAOK1 Q7L7X3 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
KMO O15229 8/20 0.43
HTR2A P28223 5/20 0.41
HTR2C P28335 5/20 0.41
HTR2B P41595 4/20 0.41
HTR1A P08908 2/20 0.41
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
HTR1D P28221 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27593382 0.89 CHEK1 (0.57) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL3980684 0.81 HTR2A (0.47) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL28140026 0.78 KMO (0.47) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL655557 0.78 KMO (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL13727172 0.77 KMO (0.52) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL655269 0.76 KMO (0.54) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL18031893 0.76 HTR2A (0.40) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL217944 0.76 HTR2A (0.45) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL31039602 0.76 HTR2A (0.45) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL13726783 0.75 KMO (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100348196-C Benzotriaza * as gastrin and cholecystokinin receptor ligands BLACK JAMES FOUNDATION (GB) 2007-11-14 CN disclosed
CN-1585643-A Benzotriazepines as gastrin and cholecystokinin receptor ligands BLACK JAMES FOUNDATION (GB) 2005-02-23 CN disclosed