SCHEMBL27612974

SCHEMBL27612974

Nc1cccc(-c2ccc(CCN3CCN(CC(C(=O)C(CN4CCN(CCc5ccc(-c6cccc(N)n6)cc5)CC4)c4ccccc4)c4ccccc4)CC3)cc2)n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 7/20 0.70
NOS3 P29474 6/20 0.70
CHRM2 P08172 1/20 0.67
CHRM4 P08173 1/20 0.67
HTR2A P28223 4/20 0.52
HTR1A P08908 2/20 0.52
DRD2 P14416 2/20 0.52
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
ASIC3 Q9UHC3 1/20 0.40
CHRM3 P20309 1/20 0.39
HTR2C P28335 3/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR2B P41595 1/20 0.38
DRD4 P21917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27594363 0.91 NOS1 (0.63) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27554919 0.91 NOS1 (0.63) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27549058 0.91 NOS1 (0.66) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27594375 0.89 NOS1 (0.63) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL6620008 0.86 NOS1 (0.74) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27612980 0.85 NOS1 (0.73) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL6618730 0.85 NOS1 (0.76) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27471830 0.85 NOS1 (0.49) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL27470928 0.85 NOS1 (0.50) NOS1NOS3CHRM2CHRM4HTR2A
SCHEMBL6618161 0.83 NOS1 (1.00) NOS1NOS3CHRM2CHRM4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1617743-A New pharmaceutical combinations for nos inhibitors PFIZER PROD INC (US) 2005-05-18 CN claimed
CN-1617743-A New pharmaceutical combinations for nos inhibitors PFIZER PROD INC (US) 2005-05-18 CN disclosed