SCHEMBL27614967

SCHEMBL27614967

CCc1ccccc1C(=O)c1sc(NCCCOS(=O)(=O)c2cccs2)nc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.40
RAB9A P51151 4/20 0.40
ALDH1A1 P00352 7/20 0.39
KDM4E B2RXH2 5/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSD17B10 Q99714 2/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
HPGD P15428 2/20 0.38
CLK2 P49760 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CDK9 P50750 1/20 0.37
LIMK1 P53667 1/20 0.37
CDK5 Q00535 1/20 0.37
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
DYRK1B Q9Y463 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14421756 0.86 NPY5R (0.45) NPC1ALDH1A1KDM4EKMT2AMEN1
SCHEMBL27614994 0.83 SMN1; SMN2 (0.43) NPC1RAB9AALDH1A1KDM4EKMT2A
SCHEMBL5570000 0.78 NPC1 (0.48) NPC1RAB9AALDH1A1KDM4EKMT2A
SCHEMBL27596188 0.76 NPY5R (0.40) NPC1RAB9AALDH1A1KDM4EKMT2A
SCHEMBL5569998 0.76 NPC1 (0.48) NPC1RAB9AALDH1A1KDM4EKMT2A
SCHEMBL27677959 0.76 NPC1 (0.50) NPC1RAB9AALDH1A1KDM4EKMT2A
SCHEMBL27614917 0.75 F2 (0.37) ALDH1A1KDM4EHSD17B10MAPK1
SCHEMBL5564500 0.73 LCK (0.43) NPC1RAB9AKMT2ACLK2GSK3A
SCHEMBL14421688 0.73 SCN1A (0.43) NPC1ALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL27614922 0.71 MAPK13 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN disclosed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN disclosed