SCHEMBL27616637

SCHEMBL27616637

c1ccc(CN2CCC(Oc3ccc4cocc4c3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 5/20 0.63
ROCK2 O75116 3/20 0.63
CCR2 P41597 2/20 0.63
HRH3 Q9Y5N1 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.56
GAA P10253 1/20 0.56
MAOA P21397 1/20 0.55
MAOB P27338 1/20 0.55
OPRK1 P41145 1/20 0.55
ACHE P22303 1/20 0.48
PARP1 P09874 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11068503 0.88 ROCK1 (0.70) ROCK1ROCK2CCR2HRH3SMN1; SMN2
Hydrochloric Acid SCHEMBL11066763 0.87 ROCK1 (0.68) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL11066614 0.84 ROCK1 (0.64) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL12192827 0.83 ROCK1 (0.76) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL10608943 0.81 ROCK1 (0.66) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL4855546 0.79 HRH3 (0.74) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL10605870 0.79 HRH1 (0.66) ROCK1ROCK2CCR2HRH3SMN1; SMN2
Hydrochloric Acid SCHEMBL10609013 0.78 HRH1 (0.65) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL5639760 0.77 ROCK2 (1.00) ROCK1ROCK2CCR2HRH3SMN1; SMN2
SCHEMBL8393625 0.77 HRH3 (0.71) ROCK1ROCK2CCR2HRH3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1639152-A Pyrrole-2, 5-dione derivatives and their use as GSK-3 inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed