SCHEMBL27620344

SCHEMBL27620344

O=COCCc1cc(Cl)ccn1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
S1PR4 O95977 3/20 0.33
PDE8A O60658 1/20 0.33
CCR1 P32246 1/20 0.33
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
FERMT2 Q96AC1 1/20 0.31
NR4A2 P43354 2/20 0.31
SOS2 Q07890 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27620343 0.98 CYP1A2 (0.33) CYP1A2ALDH1A1MAPTL3MBTL1S1PR4
SCHEMBL5541944 0.90 KCNH2 (0.36) CYP1A2ALDH1A1MAPTL3MBTL1S1PR4
SCHEMBL27777586 0.83 KDM4E (0.36) ALDH1A1CCNCCDK8KDM4E
SCHEMBL14680553 0.83 MAPT (0.35) CYP1A2ALDH1A1MAPTL3MBTL1S1PR4
Hydrochloric Acid SCHEMBL28293574 0.81 MAPT (0.34) CYP1A2ALDH1A1MAPTL3MBTL1S1PR4
SCHEMBL23639466 0.77 CYP1A2 (0.37) CYP1A2ALDH1A1MAPTL3MBTL1PDE8A
SCHEMBL27667500 0.75 DAO (0.33) L3MBTL1KDM4E
SCHEMBL5252807 0.74 HRH1 (0.50) CYP1A2ALDH1A1KDM4EHPGD
SCHEMBL5541218 0.73 RECQL (0.49)
SCHEMBL3363951 0.73 ALDH1A1 (0.38) CYP1A2ALDH1A1MAPTL3MBTL1PDE8A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102015636-B Azetidines and cyclobutanes as histamine H3 receptor antagonists EVOTEC NEUROSCIENCES GMBH 2014-08-13 CN disclosed
CN-101454311-B Salt of phenoxypyridine derivative, crystal thereof and process for producing the same EISAI R&D MAN CO LTD 2013-03-27 CN disclosed
CN-102015636-A Azetidines and cyclobutanes as histamine H3 receptor antagonists EVOTEC NEUROSCIENCES GMBH 2011-04-13 CN disclosed
CN-1711347-B Use of metal complex compounds as oxidation catalysts CIBA SC HOLDING AG 2010-05-26 CN disclosed
CN-101454311-A Salt of phenoxypyridine derivative, crystal thereof and process for producing the same EISAI R&D MAN CO LTD (JP) 2009-06-10 CN disclosed
CN-101163693-A Antibacterial piperidine derivatives ASTRAZENECA AB (SE) 2008-04-16 CN disclosed
CN-101098753-A Use of metal complexes with bispyridylpyrimidine or bispyridyltriazine ligands as catalysts for reactions with peroxides for bleaching coloured stains on hard surfaces CIBA SC HOLDING AG (CH) 2008-01-02 CN disclosed
CN-1711347-A Use of metal complex compounds as oxidation catalysts CIBA SC HOLDING AG (CH) 2005-12-21 CN disclosed