SCHEMBL27623947

SCHEMBL27623947

O=C(c1cccc(-c2cccs2)c1)c1cccc(-c2cccs2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 2/20 0.55
HTR1A P08908 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CCKAR P32238 1/20 0.50
HTR5A P47898 1/20 0.50
HDAC3 O15379 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
ABL1 P00519 2/20 0.47
BCR P11274 2/20 0.47
ERN1 O75460 1/20 0.46
PRMT6 Q96LA8 1/20 0.46
KCNH2 Q12809 1/20 0.46
ATM Q13315 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
HTR2A P28223 1/20 0.44
FYN P06241 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12551759 0.89 KAT6A (0.49) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL940399 0.87 KAT6A (0.57) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL31222146 0.87 KAT6A (0.57) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL4052204 0.86 FYN (0.57) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL4559856 0.86 AR (0.52) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL28231048 0.85 ABL1 (0.55) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL27905638 0.84 KAT6A (0.58) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL29860752 0.83 KAT6A (0.50) KAT6AHTR1AADORA3CCKARHTR5A
SCHEMBL27605045 0.82 ABL1 (0.55) HDAC2ABL1BCRERN1L3MBTL1
SCHEMBL6802813 0.82 HTR1A (0.54) KAT6AHTR1AADORA3CCKARHTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed