SCHEMBL27625366

SCHEMBL27625366

CCOC(=O)C(C)(C)c1ccc(C(N)=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 3/20 0.50
F2 P00734 2/20 0.47
F10 P00742 2/20 0.47
PLG P00747 2/20 0.47
PRSS1 P07477 1/20 0.47
MAPT P10636 1/20 0.46
CNR2 P34972 5/20 0.46
RORC P51449 1/20 0.45
EPHX2 P34913 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
MAPK1 P28482 2/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
PARP4 Q9UKK3 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447291 0.85 CA1 (0.58) MAPTCNR2MAPK1LMNACYP1A2
SCHEMBL6040918 0.85 CNR2 (0.47) F2F10PLGPRSS1MAPT
SCHEMBL13477414 0.84 PARP1 (0.47) F2F10PLGPRSS1MAPT
SCHEMBL27980232 0.83 CNR2 (0.48) F2F10PLGPRSS1MAPT
SCHEMBL397134 0.83 CYP1A2 (0.53) F2F10PLGPRSS1MAPT
SCHEMBL6279399 0.82 CNR2 (0.58) F2F10PLGPRSS1MAPT
Hydrochloric Acid SCHEMBL12273902 0.81 CYP1A2 (0.51) F2F10PLGPRSS1MAPT
SCHEMBL23582988 0.81 PARP10 (0.50) PARP10MAPTCNR2EPHX2NR1H4
SCHEMBL4115523 0.81 CNR2 (0.53) CNR2RORCLMNACYP3A4ALDH1A1
SCHEMBL24172235 0.81 GSK3B (0.51) F2F10PLGPRSS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102174024-B 2,4-pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS INC 2015-02-11 CN disclosed
CN-102174024-A 2,4-pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS INC 2011-09-07 CN disclosed
CN-1625400-B 2, 4-pyrimidinediamine compounds and uses thereof RIGEL PHARMACEUTICALS INC 2011-04-13 CN disclosed
CN-1625400-A 2, 4-pyrimidinediamine compounds and uses thereof RIGEL PHARMACEUTICALS INC (US) 2005-06-08 CN disclosed