SCHEMBL27636593

SCHEMBL27636593

[c]1cc(-c2cncs2)co1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.37
DYRK2 Q92630 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
MAPT P10636 1/20 0.32
HDAC8 Q9BY41 1/20 0.31
CD38 P28907 4/20 0.31
CHEK1 O14757 1/20 0.31
CHEK2 O96017 1/20 0.31
PRMT5 O14744 1/20 0.30
WDR77 Q9BQA1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL571374 0.68 HDAC8 (0.50) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL17701204 0.67 DYRK1A (0.41) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL17701181 0.67 DYRK1A (0.41) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL6260 0.65 DYRK1A (0.43) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL18437163 0.65 HDAC8 (0.31) DYRK1AHDAC8
SCHEMBL48894 0.64 DYRK1A (0.55) DYRK1ADYRK2DYRK1BMAPTCD38
SCHEMBL1872880 0.64 DYRK1A (0.55) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL3609293 0.64 DYRK1A (0.46) DYRK1ADYRK2DYRK1BMAPTCD38
SCHEMBL17701217 0.64 DYRK1A (0.46) DYRK1ADYRK2DYRK1BMAPTHDAC8
SCHEMBL17701233 0.63 DYRK1A (0.41) DYRK1ADYRK2DYRK1BMAPTHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1829721-A Spiro '1-azabicyclo' 2.2.2! octan-3,5'-oxazolidin - 2'-one! derivatives with affinity to the alpha7 nicotinic acetylcholine receptor ASTRAZENECA AB (SE) 2006-09-06 CN claimed
CN-1829721-A Spiro '1-azabicyclo' 2.2.2! octan-3,5'-oxazolidin - 2'-one! derivatives with affinity to the alpha7 nicotinic acetylcholine receptor ASTRAZENECA AB (SE) 2006-09-06 CN disclosed