SCHEMBL27639730

SCHEMBL27639730

CC(C)(C)OC(=O)C1COc2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.50
MAOB P27338 3/20 0.50
ROCK2 O75116 2/20 0.45
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1519495 0.85 TP53 (0.55) TP53MAOBROCK2ADORA2AADORA1
SCHEMBL17594551 0.82 TP53 (0.44) TP53MAOBROCK2
SCHEMBL24239390 0.82 TP53 (0.44) TP53MAOBROCK2
SCHEMBL5015706 0.82 ESR2 (0.49) TP53MAOB
SCHEMBL17443379 0.81 TP53 (0.55) TP53MAOB
SCHEMBL7357666 0.81 EPHX2 (0.43)
SCHEMBL31277829 0.81 ROCK2 (0.48) TP53ROCK2HDAC1HDAC2
SCHEMBL28685553 0.81 ROCK2 (0.48) TP53ROCK2HDAC1HDAC2
SCHEMBL10205890 0.80 TP53 (0.56) TP53MAOBROCK2ADORA2AADORA1
SCHEMBL4980691 0.78 TP53 (0.53) TP53MAOBROCK2ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601150-A Fused bicyclic RAF inhibitors and methods of use thereof 爵士制药爱尔兰有限公司 2023-08-15 CN disclosed
CN-102159562-A Chromene modulators of chemokine receptor activity BRISTOL MYERS SQUIBB CO 2011-08-17 CN disclosed
CN-1863799-B Chromancarboxylic acid derivatives for the treatment of diabetes and lipid disorders SK CORP 2010-09-22 CN disclosed
CN-1863799-A Chromancarboxylic acid derivatives for the treatment of diabetes and lipid disorders SK CORP (KR) 2006-11-15 CN disclosed