SCHEMBL27641069

SCHEMBL27641069

CC(C)(C)C(=O)ON1CCN(c2cccc3c2CCN(S(=O)(=O)c2ccccc2)C3)CC1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.57
DRD3 P35462 7/20 0.57
DRD2 P14416 5/20 0.53
AKR1C3 P42330 8/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
AKR1C1 Q04828 2/20 0.46
AKR1C2 P52895 1/20 0.45
GAA P10253 1/20 0.45
GFER P55789 1/20 0.45
LMNA P02545 2/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204205 0.86 HTR6 (0.57) HTR6DRD3DRD2AKR1C3MEN1
SCHEMBL5200724 0.83 HTR6 (0.81) HTR6DRD3DRD2AKR1C3MEN1
SCHEMBL6179536 0.82 HTR6 (0.62) HTR6DRD3DRD2AKR1C3MEN1
SCHEMBL5204332 0.77 HTR6 (0.82) HTR6DRD3DRD2AKR1C3MEN1
Trifluoroacetic Acid SCHEMBL5205906 0.77 HTR6 (0.69) HTR6DRD3DRD2AKR1C3MEN1
Tert-Butyl Formate SCHEMBL27641071 0.77 HTR6 (0.66) HTR6DRD3DRD2AKR1C3MEN1
SCHEMBL27548963 0.75 HTR6 (0.67) HTR6DRD3DRD2
SCHEMBL27707626 0.73 CD44 (0.39) HTR6MEN1KMT2A
SCHEMBL27568637 0.73 HTR6 (0.47) HTR6DRD2MEN1KMT2A
SCHEMBL5200784 0.70 HTR6 (0.62) HTR6DRD3DRD2LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100395237-C 2,5- and 2,6-substituted tetrahydroisoquinolines for use as 5-HT6 modulators ROCHE PALO ALTO LLC (CH) 2008-06-18 CN disclosed
CN-1756550-A 2,5- and 2,6-substituted tetrahydroisoquinolines for use as 5-HT6 modulators ROCHE PALO ALTO LLC (CH) 2006-04-05 CN disclosed