SCHEMBL27644693

SCHEMBL27644693

CCOc1cc(OCC)c(C(C)C(C)CC(N)C(=O)O)c(OCC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.41
PTGS2 P35354 4/20 0.40
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2C Q14957 1/20 0.35
NPC1 O15118 1/20 0.35
USP2 O75604 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC1A3 P43003 3/20 0.35
SLC1A2 P43004 3/20 0.35
SLC1A1 P43005 2/20 0.35
CREBBP Q92793 1/20 0.35
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27665388 0.87 KDM4E (0.36) PTGS2KDM4ETSHR
SCHEMBL28761438 0.87 SLC7A5 (0.39) SLC7A5PTGS2AKR1C3AKR1C2KDM4E
SCHEMBL27644071 0.86 TSHR (0.40) SLC7A5PTGS2AKR1C3AKR1C2KDM4E
SCHEMBL27665797 0.85 PTGS1 (0.43) SLC7A5PTGS2KDM4EPTGS1SLC1A3
SCHEMBL4984608 0.84 PTGS2 (0.39) PTGS2AKR1C3AKR1C2KDM4ENPC1
SCHEMBL27665757 0.84 AKR1C3 (0.45) SLC7A5PTGS2AKR1C3AKR1C2KDM4E
SCHEMBL27665424 0.83 PTGS2 (0.48) SLC7A5PTGS2AKR1C3AKR1C2SLC1A3
SCHEMBL27644278 0.82 SLC1A3 (0.39) SLC7A5PTGS2AKR1C3AKR1C2KDM4E
SCHEMBL27644343 0.82 AKR1C3 (0.45) SLC7A5PTGS2AKR1C3AKR1C2KDM4E
SCHEMBL27644290 0.81 GRIK1 (0.41) SLC7A5SLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1886363-A Amino acids with affinity for the alpha2delta-protein WARNER LAMBERT CO (US) 2006-12-27 CN claimed
CN-1886363-A Amino acids with affinity for the alpha2delta-protein WARNER LAMBERT CO (US) 2006-12-27 CN disclosed