SCHEMBL27645976

SCHEMBL27645976

O=C(O)c1ccc2[nH]c(-c3n[nH]c4ccsc34)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 10/20 0.54
LCK P06239 2/20 0.54
TXK P42681 2/20 0.54
SYK P43405 2/20 0.54
CSNK2A1 P68400 2/20 0.44
PARP1 P09874 1/20 0.44
CSNK2A2 P19784 1/20 0.44
CSNK2B P67870 1/20 0.44
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
MAP2K4 P45985 4/20 0.39
MAPK1 P28482 3/20 0.39
MAPKAPK3 Q16644 3/20 0.39
MAPK6 Q16659 3/20 0.39
HRH3 Q9Y5N1 1/20 0.38
CHEK1 O14757 1/20 0.37
CDK7 P50613 1/20 0.37
SPR P35270 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1623341 0.90 ITK (0.63) ITKLCKTXKSYKCSNK2A1
SCHEMBL1620556 0.90 ITK (0.51) ITKLCKTXKSYKCHEK1
SCHEMBL1623956 0.86 ITK (0.58) ITKLCKTXKSYKCHEK1
SCHEMBL1622112 0.80 ITK (0.55) ITKLCKTXKSYKCSNK2A1
SCHEMBL1622817 0.80 ITK (0.65) ITKLCKTXKSYK
SCHEMBL1622468 0.79 ITK (0.57) ITKLCKTXKSYKPARP1
SCHEMBL1627170 0.78 NPC1 (0.48) ITKLCKTXKSYKMAPK1
SCHEMBL1628603 0.78 ITK (0.62) ITKLCKTXKSYKCHEK1
SCHEMBL4125482 0.78 ITK (0.81) ITKMAP2K4MAPK1MAPKAPK3MAPK6
SCHEMBL1623125 0.77 ITK (0.50) ITKLCKTXKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100398545-C Thienopyrazoles AVENTIS PHARMA INC (US) 2008-07-02 CN claimed
CN-1849322-A Thienopyrazoles AVENTIS PHARMA INC (US) 2006-10-18 CN claimed