SCHEMBL27650451

SCHEMBL27650451

Cc1ccc2c(N3CCN(CCc4cccc(NC(N)=O)c4)CC3)cccc2n1

nearest known ligand 0.84

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 20/20 0.84
HTR1D P28221 20/20 0.84
HTR1B P28222 20/20 0.84
DRD2 P14416 6/20 0.84
HTR7 P34969 6/20 0.84
DRD3 P35462 6/20 0.84
KCNH2 Q12809 6/20 0.84
HTR2A P28223 5/20 0.84
HTR2C P28335 5/20 0.84
HTR2B P41595 5/20 0.84
HTR6 P50406 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6065943 0.99 HTR1A (0.83) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL3024414 0.96 HTR1A (0.78) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2883811 0.93 HTR1A (0.89) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2881424 0.93 HTR1A (0.88) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2883898 0.92 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2880857 0.91 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2882750 0.91 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2885358 0.90 HTR1A (0.98) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL27650505 0.90 HTR1A (0.77) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2881638 0.89 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN claimed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN claimed
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN disclosed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN disclosed