SCHEMBL27650657

SCHEMBL27650657

CCC(CC)c1ccc(CC(C)NCc2ccc(-c3ccc(CN4Cc5ccccc5CC4C(=O)O)s3)cc2)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 10/20 0.34
ACE2 Q9BYF1 2/20 0.34
MME P08473 2/20 0.34
MMP3 P08254 1/20 0.34
MMP8 P22894 1/20 0.34
MMP13 P45452 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
KLKB1 P03952 1/20 0.33
KLK1 P06870 1/20 0.33
ABCB11 O95342 1/20 0.33
TRPV1 Q8NER1 2/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27650545 0.88 KLKB1 (0.34) ACEACE2MMEMMP3MMP8
SCHEMBL6000208 0.83 S1PR1 (0.39) ACEMMP3MMP8MMP13ABCB11
SCHEMBL6000212 0.83 S1PR1 (0.39) ACEMMP3MMP8MMP13ABCB11
SCHEMBL6000132 0.78 NR4A2 (0.39) MMP3MMP8
SCHEMBL6000125 0.78 NR4A2 (0.39) MMP3MMP8
SCHEMBL5999897 0.72 S1PR1 (0.40) ACEMMP3MMP8MMP13
SCHEMBL5999898 0.72 S1PR1 (0.40) ACEMMP3MMP8MMP13
SCHEMBL5999041 0.66 S1PR1 (0.37) ACEMMP3MMP8MMP13
SCHEMBL5999037 0.66 S1PR1 (0.37) ACEMMP3MMP8MMP13
SCHEMBL7478005 0.64 ACE (0.49) ACEMMP3MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1780823-A Heteroaromatic pentacyclic compound and medicinal use thereof JAPAN TOBACCO INC (JP) 2006-05-31 CN claimed
CN-1780823-A Heteroaromatic pentacyclic compound and medicinal use thereof JAPAN TOBACCO INC (JP) 2006-05-31 CN disclosed