SCHEMBL27650993

SCHEMBL27650993

Nc1ncsc1CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 3/20 0.43
GABRB2 P47870 3/20 0.43
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.40
GABRP O00591 2/20 0.39
GABRD O14764 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB1 P18505 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA3 P34903 2/20 0.39
GABRA2 P47869 2/20 0.39
GABRA4 P48169 2/20 0.39
GABRE P78334 2/20 0.39
GABRA6 Q16445 2/20 0.39
GABRG1 Q8N1C3 2/20 0.39
GABRG3 Q99928 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2208741 0.76 KDM4E (0.52) HSD17B10MEN1KMT2AALDH1A1CYP1A2
SCHEMBL27745508 0.76 GABRA5 (0.36) GABRA5GABRB2HSD17B10MEN1KMT2A
SCHEMBL28787873 0.74 GABRA5 (0.35) GABRA5GABRB2HSD17B10MEN1KMT2A
SCHEMBL13368577 0.74
SCHEMBL23229537 0.70
Formic Acid SCHEMBL31557645 0.69 KDM4E (0.32) MEN1KMT2AALDH1A1CYP1A2KDM4E
SCHEMBL27826012 0.69 GABRR1 (0.41) GABRA5GABRB2HSD17B10MEN1KMT2A
SCHEMBL27555407 0.68
SCHEMBL27895065 0.68 GABRR1 (0.39) GABRA5GABRB2HSD17B10MEN1KMT2A
SCHEMBL1082931 0.67 PTGDR2 (0.57) MEN1KMT2AALDH1A1CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105579447-A Ethynyl derivatives HOFFMANN LA ROCHE 2016-05-11 CN disclosed
CN-102209714-B Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes UNIV BASEL 2015-03-25 CN disclosed
CN-101405275-B Triazolone Derivatives EISAI R&D MAN CO LTD 2011-11-09 CN disclosed
CN-101405275-A Triazolone Derivatives EISAI R&D MAN CO LTD (JP) 2009-04-08 CN disclosed
CN-101133054-A 1, 3-thiazole-5-carboxamides useful as cancer chemotherapeutic agents BAYER PHARMACEUTICALS CORP (US) 2008-02-27 CN disclosed
CN-1902201-A Bicyclic pyrimidin-4-(3H)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (VR1) MERCK SHARP & DOHME (GB) 2007-01-24 CN disclosed