SCHEMBL2765797

SCHEMBL2765797

COc1cc(-c2cc(CO)nn2Cc2ccccc2)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 3/20 0.46
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HSD17B10 Q99714 3/20 0.46
USP2 O75604 2/20 0.46
HPGD P15428 2/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
CHEK1 O14757 1/20 0.46
NEK2 P51955 1/20 0.46
LIMK1 P53667 1/20 0.46
TYRO3 Q06418 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
SLC16A1 P53985 2/20 0.45
MCTS1 Q9ULC4 2/20 0.45
TP53 P04637 3/20 0.44
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2764392 0.88 PDE4A (0.47) SLC16A3PDE4APDE4BPDE4CPDE4D
SCHEMBL2764448 0.87 P2RX7 (0.47) SLC16A3PDE4BALDH1A1HSD17B10HPGD
SCHEMBL2763745 0.85 BCHE (0.49) PDE4APDE4BPDE4CPDE4DTP53
SCHEMBL2766860 0.82 SLC29A1 (0.50) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL2225688 0.82 SLC16A3 (0.59) SLC16A3ALDH1A1SLC16A1MCTS1LMNA
SCHEMBL2766939 0.81 FYN (0.38) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL2764186 0.78 FYN (0.40) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL2765141 0.78 TDP1 (0.54) ALDH1A1HSD17B10USP2HPGDMAPT
SCHEMBL2764588 0.77 P2RX7 (0.47) SLC16A3PDE4BALDH1A1HSD17B10HPGD
SCHEMBL3603031 0.74 PDE4B (0.45) SLC16A3PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1400515-B1 CYCLIC DIAMINE COMPOUND HAVING FIVE-MEMBERED CYCLIC GROUP KOWA CO (JP) 2010-04-14 EP disclosed
EP-1400515-A1 CYCLIC DIAMINE COMPOUND HAVING FIVE-MEMBERED CYCLIC GROUP Kowa Co., Ltd. (JP) 2004-03-24 EP disclosed
US-6472386-B1 Cyclic diamine compound with 5-membered ring groups KOWA CO., LTD. (JP) 2002-10-29 US disclosed