SCHEMBL27664665

SCHEMBL27664665

O=C(c1csc(N(C(=O)c2ccccc2Cl)c2ccc(Cl)cc2)n1)N1CC=CC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
HTR2C P28335 6/20 0.39
ALDH1A1 P00352 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TRPC3 Q13507 2/20 0.36
TRPC6 Q9Y210 2/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MGLL Q99685 1/20 0.35
SCN9A Q15858 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032645 0.90 CYP3A4 (0.40) KDM4EHTR2CRAB9ASMN1; SMN2NPC1
SCHEMBL5032533 0.88 HTR2C (0.42) KDM4EHTR2CALDH1A1RAB9ASMN1; SMN2
SCHEMBL5034664 0.87 KMT2A (0.47) KDM4EHTR2CALDH1A1RAB9ASMN1; SMN2
SCHEMBL27664672 0.87 HTR2C (0.56) KDM4EHTR2CALDH1A1RAB9ASMN1; SMN2
SCHEMBL27643396 0.85 KMT2A (0.48) HTR2CALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL5034842 0.85 HTR2C (0.46) KDM4EHTR2CALDH1A1RAB9ASMN1; SMN2
SCHEMBL5034980 0.84 KDM4E (0.47) KDM4EALDH1A1RAB9ASMN1; SMN2HPGD
SCHEMBL5034975 0.83 KDM4E (0.44) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL5032604 0.80 TRPC3 (0.42) KDM4EHTR2CALDH1A1RAB9ASMN1; SMN2
SCHEMBL5032552 0.80 NPC1 (0.45) HTR2CALDH1A1RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN claimed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN claimed
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN disclosed