SCHEMBL27664672

SCHEMBL27664672

O=C(c1csc(N(C(=O)c2ccccc2Cl)c2ccc(Cl)cc2)n1)N1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.56
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 3/20 0.41
PHGDH O43175 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
MGLL Q99685 1/20 0.40
OPRK1 P41145 1/20 0.40
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032522 0.90 HTR2C (0.48) HTR2CNPC1RAB9ASMN1; SMN2TP53
SCHEMBL5032533 0.89 HTR2C (0.42) HTR2CNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL27643396 0.89 KMT2A (0.48) HTR2CNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL5034664 0.89 KMT2A (0.47) HTR2CNPC1RAB9ASMN1; SMN2TP53
SCHEMBL27664665 0.87 KDM4E (0.40) HTR2CNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL27643378 0.86 HTR2C (0.49) HTR2CNPC1RAB9AHPGDKMT2A
SCHEMBL5034842 0.84 HTR2C (0.46) HTR2CNPC1RAB9ASMN1; SMN2TP53
SCHEMBL5034878 0.81 KMT2A (0.48) RAB9ASMN1; SMN2MAPK1ALDH1A1ALOX15
SCHEMBL5034980 0.81 KDM4E (0.47) RAB9ASMN1; SMN2TP53KDM4EHPGD
SCHEMBL5032552 0.81 NPC1 (0.45) HTR2CNPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN claimed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN claimed
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN disclosed