SCHEMBL27668014

SCHEMBL27668014

NCCN1CCCCC1.O=C1CCN(C2CCCCC2c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 17/20 0.54
SLC6A5 Q9Y345 8/20 0.44
OPRM1 P35372 6/20 0.43
KCNH2 Q12809 1/20 0.43
OPRL1 P41146 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5562017 0.84 SLC6A9 (0.54) SLC6A9SLC6A5OPRM1KCNH2OPRL1
SCHEMBL5556937 0.84 SLC6A9 (0.54) SLC6A9SLC6A5OPRM1KCNH2OPRL1
SCHEMBL8286207 0.84 SLC6A9 (0.54) SLC6A9SLC6A5OPRM1KCNH2OPRL1
SCHEMBL5556935 0.84 SLC6A9 (0.54) SLC6A9SLC6A5OPRM1KCNH2OPRL1
SCHEMBL10740876 0.73 SMN1; SMN2 (0.57) SLC6A9SLC6A5OPRM1
SCHEMBL5556733 0.70 SLC6A9 (1.00) SLC6A9SLC6A5OPRM1OPRL1
SCHEMBL5556730 0.70 SLC6A9 (1.00) SLC6A9SLC6A5OPRM1OPRL1
SCHEMBL27625961 0.68 SLC18A3 (0.51) SLC6A9SLC6A5OPRM1KCNH2
SCHEMBL27719321 0.67 SLC6A9 (0.50) SLC6A9SLC6A5OPRM1KCNH2OPRL1
SCHEMBL13119224 0.66 HPGD (0.53) SLC6A9SLC6A5OPRM1KCNH2OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100467468-C Triaza-spiropiperidine derivatives for use as GLYT-1 inhibitors in the treatment of neurological and neuropsychiatric disorders HOFFMANN LA ROCHE (CH) 2009-03-11 CN disclosed
CN-1871238-A Triaza-spiropiperidine derivatives for use as GLYT-1 inhibitors in the treatment of neurological and neuropsychiatric disorders HOFFMANN LA ROCHE (CH) 2006-11-29 CN disclosed