SCHEMBL27670566

SCHEMBL27670566

Cc1ccc2c(N3CCN(CCc4cccc(N(C(N)=O)C(C)C)c4)CC3)cccc2n1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.72
HTR1D P28221 18/20 0.72
HTR1B P28222 18/20 0.72
CYP2C9 P11712 2/20 0.63
DRD2 P14416 6/20 0.63
HTR7 P34969 6/20 0.63
DRD3 P35462 6/20 0.63
KCNH2 Q12809 5/20 0.63
HTR2A P28223 5/20 0.63
HTR2C P28335 5/20 0.63
HTR2B P41595 5/20 0.63
HTR6 P50406 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27650478 0.92 HTR1A (0.68) HTR1AHTR1DHTR1BCYP2C9DRD2
SCHEMBL4938096 0.89 HTR1A (0.76) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27650639 0.88 HTR1A (0.75) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27670565 0.85 HTR1A (0.71) HTR1AHTR1DHTR1BCYP2C9DRD2
SCHEMBL3995158 0.85 HTR1A (0.88) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27650509 0.84 HTR1A (0.69) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27650486 0.84 HTR1A (0.69) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27670564 0.84 HTR1A (0.69) HTR1AHTR1DHTR1BCYP2C9DRD2
SCHEMBL2895887 0.84 HTR1A (1.00) HTR1AHTR1DHTR1BCYP2C9DRD2
Hydrochloric Acid SCHEMBL27670561 0.83 HTR1A (0.68) HTR1AHTR1DHTR1BCYP2C9DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN disclosed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN disclosed