SCHEMBL27674073

SCHEMBL27674073

CCOC(=O)Nc1nc(C(F)(F)F)c[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KMT2A Q03164 2/20 0.42
NPC1 O15118 2/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 2/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
KCNQ3 O43525 2/20 0.40
KCNQ2 O43526 2/20 0.40
KCNQ4 P56696 1/20 0.40
KCNQ5 Q9NR82 1/20 0.40
GAA P10253 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.38
MAPT P10636 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27564437 0.79 KMT2A (0.44) ALDH1A1KMT2APOLBKDM4EKCNQ3
SCHEMBL1970751 0.76 KDM4E (0.43) ALDH1A1KMT2AKDM4ECYP1A2HPGD
SCHEMBL27584490 0.74 MAPT (0.44) ALDH1A1KMT2ANPC1POLBKDM4E
SCHEMBL27564880 0.72 MAPT (0.42) ALDH1A1KMT2ANPC1POLBKDM4E
SCHEMBL28750125 0.71 ALDH1A1 (0.49) ALDH1A1NPC1POLBKDM4EGLA
SCHEMBL27584308 0.71 HTT (0.44) ALDH1A1KMT2ANPC1POLBKDM4E
SCHEMBL27564521 0.71 ALDH1A1 (0.38) ALDH1A1KMT2AGAACYP1A2CYP2C9
SCHEMBL10717894 0.71 ALDH1A1 (0.46) ALDH1A1KMT2APOLBKCNQ3KCNQ2
SCHEMBL20078909 0.69 KMT2A (0.50) ALDH1A1KMT2ANPC1POLBKDM4E
SCHEMBL8392811 0.69 KMT2A (0.46) ALDH1A1KMT2APOLBKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006063-B Five-membered heterocycles useful as serine protease inhibitors. BRISTOL MYERS SQUIBB CO 2013-07-17 CN disclosed
CN-101006063-A Five-membered heterocycles useful as serine protease inhibitors. BRISTOL MYERS SQUIBB CO (US) 2007-07-25 CN disclosed