SCHEMBL27675002

SCHEMBL27675002

O=C(O)N1CCN(C(C#Cc2cccc(Cl)c2)c2ccccc2Cl)CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HTT P42858 2/20 0.47
LMNA P02545 1/20 0.47
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CACNA2D1 P54289 10/20 0.42
CACNA1B Q00975 10/20 0.42
CACNB1 Q02641 10/20 0.42
CACNA1C Q13936 4/20 0.42
CACNA1G O43497 3/20 0.40
CNR1 P21554 5/20 0.39
CNR2 P34972 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27655169 0.89 MAPT (0.46) MAPTALDH1A1HTTLMNAKDM4E
SCHEMBL27655175 0.87 CACNA2D1 (0.46) MAPTALDH1A1HTTLMNACACNA2D1
SCHEMBL5710807 0.86 GRM5 (0.56) MAPTALDH1A1HTTLMNA
SCHEMBL27674992 0.85 MAPT (0.42) MAPTALDH1A1HTTLMNACACNA2D1
SCHEMBL27675173 0.81 MEN1 (0.44) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1G
SCHEMBL27655170 0.80 CACNA2D1 (0.39) MAPTALDH1A1HTTLMNACACNA2D1
SCHEMBL27655174 0.79
SCHEMBL27655166 0.78 MEN1 (0.41) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1G
SCHEMBL27675030 0.78 CACNA2D1 (0.44) ALDH1A1LMNASMN1; SMN2CACNA2D1CACNA1B
SCHEMBL27655173 0.77 GRM5 (0.40) MAPTALDH1A1HTTCACNA2D1CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1934097-A Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists ASTRAZENECA AB (SE) 2007-03-21 CN claimed
CN-1934097-A Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists ASTRAZENECA AB (SE) 2007-03-21 CN disclosed