SCHEMBL27678917

SCHEMBL27678917

O=C(O)c1coc(CCBr)n1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.39
P2RY2 P41231 1/20 0.34
ALOX15 P16050 2/20 0.33
TSHR P16473 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ACMSD Q8TDX5 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HIF1A Q16665 1/20 0.32
PTPN1 P18031 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
FBP1 P09467 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL744062 0.85 CES1 (0.38) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL18782175 0.81 HCAR2 (0.42) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL18782173 0.81 CES1 (0.39) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL16011738 0.81 CES1 (0.39) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL15931723 0.79 HCAR2 (0.45) CES1ALOX15TSHRKDM4ETDP1
SCHEMBL742811 0.79 CES1 (0.39) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL27603649 0.77 CYP1A2 (0.46) TSHRKDM4EFBP1ALDH1A1
SCHEMBL3590995 0.77 CES1 (0.38) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL1972922 0.77 CES1 (0.38) CES1P2RY2ALOX15TSHRKDM4E
SCHEMBL1811036 0.77 CES1 (0.38) CES1P2RY2ALOX15TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1938273-B Tetrahydrocarbazoles and derivatives HOFFMAN-LA ROCHE LTD. (CH) 2011-12-14 CN disclosed
CN-1938273-A Tetrahydrocarbazoles and derivatives HOFFMANN LA ROCHE (CH) 2007-03-28 CN disclosed