SCHEMBL27697217

SCHEMBL27697217

Nc1ccc(C(=O)Nc2ccc(-n3c(C(F)(F)F)nc4ccccc43)cc2)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPC1 P48995 1/20 0.40
TRPC3 Q13507 1/20 0.40
STIM1 Q13586 1/20 0.40
ORAI1 Q96D31 1/20 0.40
GPR27 Q9NS67 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 2/20 0.39
AURKA O14965 1/20 0.39
KDR P35968 1/20 0.39
AURKB Q96GD4 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PTGS1 P23219 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
MCL1 Q07820 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27717168 0.92 MAPK1 (0.42) TRPC1TRPC3STIM1ORAI1CYP2C9
SCHEMBL2096523 0.90 NPC1 (0.50) TRPC1TRPC3STIM1ORAI1GPR27
SCHEMBL27717256 0.88 MEN1 (0.47) TRPC1TRPC3STIM1ORAI1NPC1
SCHEMBL27717099 0.88 MEN1 (0.53) MAPK1NPC1MAPTRAB9AMEN1
SCHEMBL2094733 0.85 PTGS1 (0.41) CYP2C9MAPK1MAPTAURKAKDR
SCHEMBL2093588 0.84 LMNA (0.43) TRPC1TRPC3STIM1ORAI1CYP2C9
SCHEMBL2091612 0.84 STIM1 (0.55) TRPC1TRPC3STIM1ORAI1CYP2C9
SCHEMBL10187707 0.83 MEN1 (0.44) MAPK1NPC1MAPTRAB9AAURKA
SCHEMBL2095257 0.83 CRACR2A (0.41) TRPC1TRPC3STIM1ORAI1NPC1
SCHEMBL2094439 0.82 KDM4E (0.40) CYP2C9MAPK1MAPTAURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101083985-A Compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP (US) 2007-12-05 CN claimed
CN-101083985-A Compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP (US) 2007-12-05 CN disclosed