SCHEMBL27697339

SCHEMBL27697339

CC(C(=O)C(C)c1ccc(Nc2cccc(-c3ncc(Cl)s3)c2)c(N)c1)c1ccc(Nc2cccc(-c3ncc(Cl)s3)c2)c(N)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 4/20 0.40
NPC1 O15118 2/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
DYRK3 O43781 2/20 0.36
CCNT1 O60563 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
CDK5 Q00535 2/20 0.36
DYRK1A Q13627 2/20 0.36
CDK5R1 Q15078 2/20 0.36
DYRK2 Q92630 2/20 0.36
DYRK1B Q9Y463 2/20 0.36
ROCK2 O75116 1/20 0.35
HDAC3 O15379 5/20 0.35
HDAC1 Q13547 5/20 0.35
HDAC2 Q92769 5/20 0.35
HDAC4 P56524 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27697342 0.86 ROCK1 (0.36) ROCK1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL27717206 0.85 MEN1 (0.42) ROCK1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL2652430 0.84 AKR1C3 (0.45) NPC1POLBRAB9ASMN1; SMN2GAA
SCHEMBL27717209 0.72 EPAS1 (0.40) ROCK1POLB
SCHEMBL2652297 0.71 MAPT (0.48) NPC1POLBRAB9ASMN1; SMN2
SCHEMBL27697313 0.71 FGFR1 (0.42) NPC1RAB9ASMN1; SMN2
SCHEMBL27618307 0.66 CTDSP1 (0.47) NPC1POLBRAB9ASMN1; SMN2GAA
SCHEMBL2650071 0.66 GAA (0.49) ROCK1NPC1SMN1; SMN2CDK2CDK5
SCHEMBL2667905 0.65 MAP4K4 (0.49) NPC1POLBRAB9ASMN1; SMN2DYRK3
SCHEMBL27896220 0.65 PRKCI (0.53) NPC1RAB9AHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101141958-A Benzimidazole derivatives and their use for modulating GABAAUse of receptor complexes NEUROSEARCH AS (DK) 2008-03-12 CN disclosed