SCHEMBL27697342

SCHEMBL27697342

CC(C=O)c1ccc(Nc2cccc(-c3ncc(Cl)s3)c2)c(N)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 5/20 0.36
HDAC3 O15379 5/20 0.33
HDAC4 P56524 5/20 0.33
HDAC1 Q13547 5/20 0.33
HDAC7 Q8WUI4 5/20 0.33
HDAC2 Q92769 5/20 0.33
HDAC10 Q969S8 5/20 0.33
HDAC11 Q96DB2 5/20 0.33
HDAC8 Q9BY41 5/20 0.33
HDAC6 Q9UBN7 5/20 0.33
HDAC9 Q9UKV0 5/20 0.33
HDAC5 Q9UQL6 5/20 0.33
BTK Q06187 2/20 0.33
NPC1 O15118 3/20 0.33
POLB P06746 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ROCK2 O75116 1/20 0.32
AAK1 Q2M2I8 2/20 0.32
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27697339 0.86 ROCK1 (0.40) ROCK1HDAC3HDAC4HDAC1HDAC7
SCHEMBL27717209 0.85 EPAS1 (0.40) ROCK1POLBMEN1ALDH1A1MAPT
SCHEMBL2652430 0.80 AKR1C3 (0.45) NPC1POLBRAB9ASMN1; SMN2ALDH1A1
SCHEMBL27717206 0.72 MEN1 (0.42) ROCK1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL27697316 0.70 FGFR1 (0.39) NPC1RAB9AALDH1A1
SCHEMBL27618309 0.66 CTDSP1 (0.44) NPC1POLBRAB9ASMN1; SMN2MEN1
SCHEMBL2667905 0.65 MAP4K4 (0.49) NPC1POLBRAB9ASMN1; SMN2MEN1
SCHEMBL27896222 0.65 PRKCI (0.45) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL27597646 0.63 MAPT (0.41) NPC1RAB9ASMN1; SMN2MEN1ALDH1A1
SCHEMBL15606529 0.61 CDK2 (0.43) HDAC4NPC1POLBRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101141958-A Benzimidazole derivatives and their use for modulating GABAAUse of receptor complexes NEUROSEARCH AS (DK) 2008-03-12 CN disclosed