SCHEMBL27697644

SCHEMBL27697644

COC(=O)Cc1c[nH]c2c(Cl)ncc(Br)c12

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.34
MTNR1B P49286 4/20 0.34
ALDH1A1 P00352 3/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ADRB3 P13945 1/20 0.32
KDM4E B2RXH2 2/20 0.31
GAA P10253 2/20 0.30
KDM5B Q9UGL1 1/20 0.30
MAPT P10636 2/20 0.30
HPGD P15428 2/20 0.30
TDP1 Q9NUW8 1/20 0.30
LMNA P02545 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2672681 0.84 ALDH1A1 (0.38) ALDH1A1KDM4EGAAMAPTHPGD
SCHEMBL2628871 0.75 NR4A2 (0.35)
SCHEMBL2254864 0.74 CYP2D6 (0.41) ALDH1A1KDM4E
SCHEMBL20422633 0.72 JAK2 (0.42) MTNR1AMTNR1BALDH1A1KDM4EMAPT
SCHEMBL2259078 0.72 SMN1; SMN2 (0.34) ALDH1A1NPC1RAB9AKDM4EGAA
SCHEMBL9755930 0.71 CSNK2A2 (0.48) MTNR1AMTNR1BALDH1A1NPC1RAB9A
SCHEMBL9937273 0.70 LRRK2 (0.47) MTNR1AMTNR1BALDH1A1NPC1RAB9A
SCHEMBL2255704 0.70 CSNK2A2 (0.35) ALDH1A1NPC1RAB9AMAPTHPGD
SCHEMBL3992292 0.70 CFB (0.32)
SCHEMBL12751060 0.69 KDM5A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101018781-A Bicyclic N-anilide spirolactam CGRP receptor antagonists MERCK & CO INC (US) 2007-08-15 CN disclosed