SCHEMBL27698459

SCHEMBL27698459

CNc1nc(N)nc2cc(-c3ccccc3C(C)C=O)ccc12

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.43
PTPN1 P18031 11/20 0.40
APP P05067 1/20 0.40
NLRP3 Q96P20 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4511008 0.87 DHFR (0.51) DHFRPTPN1APPNLRP3
SCHEMBL27698454 0.84 DHFR (0.43) DHFRPTPN1APPNLRP3CYP1A2
SCHEMBL4511017 0.81 DHFR (0.47) DHFRPTPN1APPNLRP3CYP1A2
SCHEMBL4519688 0.80 DHFR (0.52) DHFRPTPN1APPNLRP3CYP1A2
SCHEMBL4515183 0.78 PTPN1 (0.59) DHFRPTPN1CYP1A2CYP3A4CYP2D6
SCHEMBL4524948 0.78 DHFR (0.48) DHFRPTPN1APPNLRP3
SCHEMBL4511415 0.78 DHFR (0.51) DHFRPTPN1APPNLRP3CYP1A2
SCHEMBL4529705 0.77 PTPN1 (0.60) DHFRPTPN1APPNLRP3
SCHEMBL4526439 0.77 DHFR (0.50) DHFRPTPN1NLRP3
SCHEMBL4524950 0.77 PTPN1 (0.60) DHFRPTPN1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101056865-A Aminoquinazolines compounds HOFFMANN LA ROCHE (CH) 2007-10-17 CN claimed
CN-101056865-A Aminoquinazolines compounds HOFFMANN LA ROCHE (CH) 2007-10-17 CN disclosed