SCHEMBL27699404

SCHEMBL27699404

Brc1ccc(-c2cn(-c3cccnc3)cn2)o1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.51
CYP2E1 P05181 4/20 0.51
CYP3A4 P08684 3/20 0.42
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
RIPK2 O43353 1/20 0.40
NLRP3 Q96P20 1/20 0.38
CYP2C9 P11712 2/20 0.35
CYP2B6 P20813 2/20 0.35
CYP2C19 P33261 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
TP53 P04637 2/20 0.34
PKM P14618 2/20 0.34
POLB P06746 2/20 0.34
GRM5 P41594 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699382 0.81 CYP2A6 (0.48) CYP2A6CYP2E1CYP3A4RIPK2CYP2C9
SCHEMBL27699265 0.79 CYP2A6 (0.46) CYP2A6CYP2E1CYP3A4ALDH1A1MAPT
SCHEMBL20259879 0.75 CYP2A6 (0.65) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL27719861 0.74 CYP2A6 (0.56) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL27719999 0.74 CYP2A6 (0.52) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL27699427 0.74 CYP2A6 (0.59) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL15825417 0.70 CYP2A6 (0.55) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL27719858 0.69 CYP2A6 (0.57) CYP2A6CYP2E1CYP3A4RIPK2CYP2C9
SCHEMBL2835686 0.69 CYP2A6 (0.52) CYP2A6CYP2E1CYP3A4RAB9ANPC1
SCHEMBL27699234 0.69 CYP2A6 (0.52) CYP2A6CYP2E1CYP3A4RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101166735-A Novel oxadiazole derivatives and their medical use NEUROSEARCH AS (DK) 2008-04-23 CN disclosed