SCHEMBL27699265

SCHEMBL27699265

O=[N+]([O-])c1ccc(-c2cn(-c3cccnc3)cn2)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.46
CYP2E1 P05181 3/20 0.46
LMNA P02545 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
RIPK2 O43353 1/20 0.39
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
ABL1 P00519 1/20 0.38
NTRK1 P04629 1/20 0.38
FYN P06241 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699256 0.85 CHEK1 (0.40) LMNACHEK1AURKADAPK3JAK2
SCHEMBL27699228 0.82 CHEK1 (0.38) LMNANFKB1NFKB2RELACHEK1
SCHEMBL27719895 0.80 CYP2A6 (0.45) CYP2A6CYP2E1RIPK2ABL1CYP3A4
SCHEMBL27699404 0.79 CYP2A6 (0.51) CYP2A6CYP2E1LMNARIPK2ABL1
SCHEMBL27699405 0.78 HPGD (0.40) LMNACHEK1AURKADAPK3JAK2
SCHEMBL27699429 0.77 TLR2 (0.52) CYP2A6CYP2E1LMNARIPK2CYP3A4
SCHEMBL27699382 0.76 CYP2A6 (0.48) CYP2A6CYP2E1RIPK2CYP3A4CYP2C9
SCHEMBL28772169 0.76 KDM4E (0.50) CYP2A6CYP2E1LMNARIPK2FGFR1
SCHEMBL17632576 0.75 CYP2A6 (0.56) CYP2A6CYP2E1RIPK2CYP3A4KDM4E
SCHEMBL27719706 0.75 KEAP1 (0.51) CYP2A6CYP2E1ABL1MAPTPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101166735-A Novel oxadiazole derivatives and their medical use NEUROSEARCH AS (DK) 2008-04-23 CN disclosed