SCHEMBL27699580

SCHEMBL27699580

c1ccc2nc(Nc3cc4ccccc4[nH]3)ncc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.45
ROCK1 Q13464 1/20 0.41
S1PR3 Q99500 1/20 0.41
ACVR1 Q04771 1/20 0.39
KDR P35968 3/20 0.37
PDE10A Q9Y233 1/20 0.37
FDPS P14324 1/20 0.36
PCSK9 Q8NBP7 1/20 0.36
PDE2A O00408 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
HTR3A P46098 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36
TOP2A P11388 1/20 0.36
AOC3 Q16853 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6467426 0.78 MAP3K5 (0.54) MAP3K5ROCK1S1PR3ACVR1KDR
SCHEMBL27075383 0.76 AOC3 (0.52) KDRNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL9921201 0.74 MAP3K5 (0.46) MAP3K5ROCK1S1PR3ACVR1PDE10A
SCHEMBL167891 0.72 MAP3K5 (0.60) MAP3K5ROCK1KDRNPC1MAPT
SCHEMBL31381352 0.72 MAP3K5 (0.60) MAP3K5ROCK1KDRNPC1MAPT
Benzene SCHEMBL28188863 0.72 MAP3K5 (0.60) MAP3K5ROCK1KDRNPC1MAPT
SCHEMBL27770482 0.72 MAP3K5 (0.60) MAP3K5ROCK1KDRNPC1MAPT
SCHEMBL22725711 0.71 ROCK1 (0.45) MAP3K5ROCK1KDRHTR3AMAPT
SCHEMBL1054022 0.71 ROCK1 (0.51) MAP3K5ROCK1KDRHTR3AFGFR1
Hydrochloric Acid SCHEMBL8807679 0.70 MAP3K5 (0.58) MAP3K5ROCK1KDRNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101171245-A Indolylamino quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2008-04-30 CN disclosed
CN-101171245-A Indolylamino quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2008-04-30 CN disclosed