SCHEMBL2770128

SCHEMBL2770128

Cc1cc(CN(C)c2ccc(OCc3c(C(C)C)cnn3-c3ccccc3OC(F)(F)F)cc2Cl)ccc1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.41
TRPM8 Q7Z2W7 7/20 0.37
MCHR1 Q99705 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770610 0.94 TRPM8 (0.38) NR1H4TRPM8MCHR1
SCHEMBL2773384 0.87 TRPM8 (0.40) NR1H4TRPM8
SCHEMBL2771847 0.87 NR1H4 (0.41) NR1H4TRPM8MCHR1
SCHEMBL2770027 0.85 NR1H4 (0.56) NR1H4MCHR1
SCHEMBL2770975 0.85 NR1H4 (0.44) NR1H4TRPM8
SCHEMBL2770584 0.81 NR1H4 (0.54) NR1H4MCHR1
SCHEMBL2773939 0.80 NR1H4 (0.52) NR1H4MCHR1
SCHEMBL2772608 0.79 PTPN1 (0.35) NR1H4TRPM8
SCHEMBL2772254 0.78 TRPM8 (0.44) NR1H4TRPM8
SCHEMBL2771742 0.78 NR1H4 (0.43) NR1H4TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed