SCHEMBL27701741

SCHEMBL27701741

O=C(S)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCD O00767 7/20 0.59
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
HTR2B P41595 1/20 0.58
MAPK14 Q16539 1/20 0.58
MGLL Q99685 1/20 0.54
GBA1 P04062 1/20 0.54
HSD11B1 P28845 1/20 0.50
NPY2R P49146 1/20 0.49
P2RX7 Q99572 1/20 0.48
TSHR P16473 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4262448 0.86 CYP2C9 (0.63) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL14172993 0.84 SCD (0.59) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL13983799 0.84 SCD (0.62) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL12894564 0.84 SCD (0.59) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL10304326 0.84 CYP2C9 (0.60) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL27701738 0.83 CYP2C9 (0.60) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL2006284 0.83 CYP2C9 (0.59) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL2820604 0.82 SCD (0.58) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL2821970 0.82 MGLL (0.58) SCDCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL4716887 0.82 SCD (0.56) SCDCYP2C9CYP2C19HTR2BMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101083982-A Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes XENON PHARMACEUTICALS INC (CA) 2007-12-05 CN disclosed