SCHEMBL2770534

SCHEMBL2770534

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1COc1ccc(CC(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 16/20 0.56
PPARD Q03181 8/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.43
FFAR1 O14842 2/20 0.40
PDGFRA P16234 1/20 0.39
S1PR1 P21453 1/20 0.39
ROCK1 Q13464 1/20 0.39
S1PR5 Q9H228 1/20 0.39
LIFR P42702 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774998 0.94 NR1H4 (0.55) NR1H4PPARDPTGDR2FFAR1PDGFRA
SCHEMBL2771465 0.90 NR1H4 (0.64) NR1H4PPARDLIFR
SCHEMBL2773870 0.89 NR1H4 (0.55) NR1H4PPARDFFAR1
SCHEMBL2787707 0.88 NR1H4 (0.59) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2773502 0.88 NR1H4 (0.54) NR1H4PPARD
SCHEMBL2770317 0.87 NR1H4 (0.68) NR1H4LIFR
SCHEMBL2773817 0.85 NR1H4 (0.54) NR1H4FFAR1
SCHEMBL2773824 0.85 NR1H4 (0.56) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2771269 0.84 NR1H4 (0.56) NR1H4PPARDFFAR1PDGFRAS1PR1
SCHEMBL2772145 0.84 NR1H4 (0.51) NR1H4PPARDFFAR1LIFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed