SCHEMBL2772145

SCHEMBL2772145

CCS(C)(c1ccc(CC(=O)O)cc1)c1ccc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)cc1C

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 16/20 0.51
PPARD Q03181 6/20 0.40
FFAR1 O14842 4/20 0.35
LIFR P42702 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769946 0.93 NR1H4 (0.50) NR1H4PPARDFFAR1
SCHEMBL2771606 0.91 NR1H4 (0.57) NR1H4LIFR
SCHEMBL2771162 0.87 NR1H4 (0.61) NR1H4LIFR
SCHEMBL3150714 0.87 NR1H4 (0.51) NR1H4PPARDFFAR1
SCHEMBL2770911 0.84 NR1H4 (0.52) NR1H4
SCHEMBL2770534 0.84 NR1H4 (0.56) NR1H4PPARDFFAR1LIFR
SCHEMBL2773502 0.84 NR1H4 (0.54) NR1H4PPARD
SCHEMBL2773870 0.84 NR1H4 (0.55) NR1H4PPARDFFAR1
SCHEMBL2771579 0.83 NR1H4 (0.40) NR1H4PPARDFFAR1
SCHEMBL2772140 0.81 NR1H4 (0.52) NR1H4PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed