SCHEMBL27705804

SCHEMBL27705804

FC(F)(F)c1ccc(Br)c(CCBr)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.39
GSK3B P49841 1/20 0.39
IDO1 P14902 2/20 0.39
PTPN5 P54829 1/20 0.37
PIEZO1 Q92508 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
DAO P14920 4/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
TAAR1 Q96RJ0 2/20 0.34
CYBB P04839 1/20 0.34
NOX3 Q9HBY0 1/20 0.34
NOX4 Q9NPH5 1/20 0.34
NOX1 Q9Y5S8 1/20 0.34
MAPT P10636 1/20 0.33
XBP1 P17861 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18586260 0.85 IDO1 (0.39) IDO1PTPN5PIEZO1DAOTAS2R14
SCHEMBL475304 0.84 IDO1 (0.41) PTPN1GSK3BIDO1PTPN5PIEZO1
SCHEMBL29382636 0.84 IDO1 (0.41) PTPN1GSK3BIDO1PTPN5PIEZO1
SCHEMBL3410622 0.83 IDO1 (0.42) PTPN1GSK3BIDO1PIEZO1DAO
SCHEMBL4597627 0.83 PPARG (0.40) IDO1PIEZO1DAOMAPTCYP3A4
SCHEMBL18586969 0.81 IDO1 (0.37) IDO1PTPN5PIEZO1SIRT2DAO
SCHEMBL27546311 0.81 IDO1 (0.54) PTPN1GSK3BIDO1PTPN5SIRT2
SCHEMBL138276 0.80 TAAR1 (0.43) IDO1PIEZO1DAOTAAR1
SCHEMBL18587132 0.80 IDO1 (0.36) IDO1PIEZO1DAOTAS2R14TAAR1
SCHEMBL18586253 0.80 CTSK (0.36) PTPN1GSK3BIDO1PIEZO1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555783-A Autotaxin inhibitors comprising a heteroaromatic ring-benzyl-amide-cycle core NOVARTIS AG 2016-05-04 CN disclosed
CN-104892532-A Synthetic process of chiral 3-substituted 1,3,4,5-tetrahydro-1,4-benzodiazepine-2-ketone UNIV CHENGDU TECHNOLOGY 2015-09-09 CN disclosed
CN-101437804-A Dibenzyl amine compounds and derivatives PFIZER PROD INC (US) 2009-05-20 CN disclosed
CN-101437803-A Dibenzyl amine derivatives as CETP inhibitors PFIZER PROD INC (US) 2009-05-20 CN disclosed
CN-101065366-A Dibenzyl amine compounds and derivatives PFIZER PROD INC (US) 2007-10-31 CN disclosed