SCHEMBL27705806

SCHEMBL27705806

CC(Br)c1cc(C(F)(F)F)ccc1Br

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 7/20 0.44
P2RX7 Q99572 1/20 0.41
HTR2A P28223 2/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
GSK3B P49841 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
SLC6A4 P31645 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PTPN5 P54829 1/20 0.34
KIF11 P52732 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MAPT P10636 1/20 0.34
XBP1 P17861 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747383 0.88 PDE2A (0.44) PDE2AHTR2AHTR2CHTR2BTAS2R14
SCHEMBL27877627 0.86 PDE2A (0.47) PDE2AP2RX7HTR2AHTR2CHTR2B
SCHEMBL6794936 0.85 PDE2A (0.59) PDE2AHTR2AHTR2CHTR2BGSK3B
SCHEMBL150245 0.85 PDE2A (0.59) PDE2AHTR2AHTR2CHTR2BGSK3B
SCHEMBL31040742 0.85 PDE2A (0.59) PDE2AHTR2AHTR2CHTR2BGSK3B
SCHEMBL31064629 0.85 PDE2A (0.59) PDE2AHTR2AHTR2CHTR2BGSK3B
Hydrochloric Acid SCHEMBL29072767 0.83 PDE2A (0.41) PDE2AHTR2AHTR2CHTR2BTAS2R14
Hydrochloric Acid SCHEMBL30117081 0.83 PDE2A (0.41) PDE2AHTR2AHTR2CHTR2BTAS2R14
SCHEMBL17698505 0.82 P2RX7 (0.47) PDE2AP2RX7HTR2AHTR2CHTR2B
SCHEMBL22717245 0.82 P2RX7 (0.47) PDE2AP2RX7HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555783-A Autotaxin inhibitors comprising a heteroaromatic ring-benzyl-amide-cycle core NOVARTIS AG 2016-05-04 CN disclosed
CN-101437804-A Dibenzyl amine compounds and derivatives PFIZER PROD INC (US) 2009-05-20 CN disclosed
CN-101437803-A Dibenzyl amine derivatives as CETP inhibitors PFIZER PROD INC (US) 2009-05-20 CN disclosed
CN-101065366-A Dibenzyl amine compounds and derivatives PFIZER PROD INC (US) 2007-10-31 CN disclosed