SCHEMBL2770735

SCHEMBL2770735

CNCCc1ccc(OCC(=O)OC)c(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.48
KDM4E B2RXH2 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
AR P10275 1/20 0.44
PPARD Q03181 3/20 0.42
PPARG P37231 2/20 0.42
PPARA Q07869 2/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL988863 0.81 PTGDR2 (0.51) PTGDR2ARPPARDPPARGPPARA
SCHEMBL2770732 0.80 AKR1C3 (0.49) PTGDR2ARPPARDPPARGPPARA
SCHEMBL988515 0.79 PTGDR2 (0.47) PTGDR2KDM4EAR
SCHEMBL23991026 0.76 KDM4E (0.43) PTGDR2KDM4ETDP1CYP1A2CYP2C19
SCHEMBL12542140 0.73 PTGDR2 (0.52) PTGDR2MEN1KMT2AMRGPRX4
SCHEMBL13770251 0.72 PTGDR2 (0.69) PTGDR2PPARDMRGPRX4
SCHEMBL3920885 0.70 TAAR1 (0.61) KDM4ECYP1A2CYP2C19MEN1KMT2A
SCHEMBL3009106 0.70 CHRM2 (0.63) PPARGPPARACYP1A2CYP2C19MEN1
SCHEMBL29580665 0.70 CHRM2 (0.63) PPARGPPARACYP1A2CYP2C19MEN1
SCHEMBL585016 0.70 KDM4E (0.68) KDM4EPPARDPPARGPPARAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010102154-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-09-10 WO disclosed